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Tasigna
nilotinib
APPROVED
Drug Profile
Modality
Small molecule
Route
Oral
Therapy Area
Oncology
Launch
2007-10-29
US LOE
2028-07-01
Peak Sales Est
$2000M
Formulations
[{"id":"tasigna-oral","doses":"50mg, 150mg, 200mg capsules","route":"Oral","setting":"PATIENT_SELF",
Companies
NVS
(ORIGINATOR)
100%
Mechanism: BCR-ABL inhibitor (STAMP)
Expert:
Specifically targets ABL myristoyl pocket (STAMP) inhibitor of BCR-ABL1
Everyday:
Blocks the abnormal protein that causes certain leukemias
Targets: ["BCR-ABL"]
Revenue History
Period
Revenue ($M)
2024
$1,680M
2025
$1,550M
Programs (1)
Indication
Stage
Key Study
Regional Status
CML
APPROVED
ENESTnd
[{"stage":"APPROVED","region":"US","approval_date":"2007-10-29"},{"stage":"APPRO
Notes
BCR-ABL inhibitor for CML. Second-gen TKI. Facing generic pressure.
Data from Supabase · Updated 2026-03-24