Padsevonil padsevonil PHASE3
Drug Profile
ModalitySmall molecule
RoutePO
Therapy AreaNeurology
Peak Sales Est$800M
Formulations[]
Companies
UCB (ORIGINATOR)100%
Mechanism: SV2A/GABAA modulator
Expert: Dual-mechanism antiepileptic that binds SV2A (similar to levetiracetam/brivaracetam) and positively modulates GABAA receptors, providing synergistic anticonvulsant activity.
Everyday: Works on two brain targets to reduce seizures - one that controls brain chemical release and one that calms nerve activity.
Targets: ["SV2A","GABA-A"]
Programs (2)
IndicationStageKey StudyRegional Status
Drug-resistant focal epilepsyPHASE3NCT04625101[]
Refractory focal epilepsyPHASE3PATTERN[]
Upcoming Catalysts (1)
Padsevonil - Drug-Resistant Epilepsy - Ph3 - Updates 2026
Notes
Dual-mechanism anticonvulsant combining SV2A modulation with GABA-A receptor positive allosteric modulation for drug-resistant epilepsy. Novel approach targeting two synergistic pathways for treatment-refractory seizures.
Data from Supabase · Updated 2026-03-24